CancerFax
TARGETED THERAPY

TYPES OF TARGETED
THERAPY DRUGS

Two patients with the same cancer type may be on completely different targeted therapy categories because their tumours have different molecular drivers. The drug follows from the mutation profile.

Reviewed by: CancerFax Medical Team, Oncology & Haematology SpecialistsLast reviewed: April 16, 20269 min read

Targeted Therapy Drug Classes at a Glance

Drug ClassMechanismRouteKey ExamplesKey Cancer Types
Tyrosine Kinase Inhibitors (TKIs)Block kinase proteins from passing growth signals inside cellsOral pillOsimertinib, alectinib, imatinibLung (EGFR/ALK), CML, GIST
Monoclonal AntibodiesBind to surface targets; block activation or recruit immune destructionIV infusionTrastuzumab, cetuximab, bevacizumabBreast, colorectal, lung
Antibody-Drug Conjugates (ADCs)Antibody delivers toxic payload directly to cancer cellsIV infusionTrastuzumab deruxtecan, T-DM1Breast, gastric, lung
PARP InhibitorsBlock DNA repair pathway BRCA-mutated cancers depend onOral pillOlaparib, niraparib, rucaparibOvarian, breast, prostate, pancreatic
CDK4/6 InhibitorsBlock proteins driving the cell division cycleOral pillPalbociclib, ribociclib, abemaciclibHR+ breast cancer
mTOR InhibitorsDisrupt pathway regulating cell growth and metabolismOral pillEverolimus, temsirolimusKidney, HR+ breast cancer
Proteasome InhibitorsDisrupt protein disposal causing lethal cell stressIV or subcutaneousBortezomib, carfilzomibMultiple myeloma

Frequently Asked Questions

    How CancerFax Helps

    CancerFax is a specialist cancer access and patient-navigation platform. We help patients and families understand their options, organise medical records, coordinate hospital communication, and support cross-border treatment planning where appropriate.

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    Medical Record Review

    We help collect and organise reports, scans, pathology, biomarker results, and treatment history for structured case review.

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    Eligibility Coordination

    We communicate with hospitals or trial teams to assess whether a case may be suitable for further screening.

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    Hospital Communication

    We support appointment coordination, document submission, translation, and direct communication with international departments.

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    Travel & Admission Support

    For international patients, we help with practical coordination — travel planning, hospital admission guidance, and local support.

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    Treatment & Trial Navigation

    If this option is not suitable, we help explore other relevant treatments, clinical trials, or advanced care pathways.

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    End-to-end Coordination

    From inquiry through to follow-up, our coordinators provide a single point of contact for the family.

    CancerFax does not guarantee treatment access, eligibility, or clinical outcome. Our role is to help patients access accurate information, structured review, and appropriate specialist pathways.

    Questions About Which Targeted Drug Class Applies to Your Diagnosis?

    CancerFax reviews your molecular profile to identify which targeted therapy categories are relevant for your specific cancer.

    This content is for informational purposes only and does not constitute medical advice. Always consult a qualified oncologist before making treatment decisions.